Efficient Synthesis of Impurity-C of Antimigraine Agent Rizatriptan Benzoate

Chinmoy Pramanik, Rahul Bhumkar, Ganesh Karhade, Pravinkumar Khairnar, Narendra Kumar Tripathy, and Mukund K. Gurjar

Org. Process Res. Dev., 2012, 16 (3), pp 507–511

DOI: 10.1021/op200284m

Practical Asymmetric Synthesis of (+)-erythro Mefloquine Hydrochloride

William P. Hems, William P. Jackson, Peter Nightingale, and Rob Bryant

Org. Process Res. Dev., 2012, 16 (3), pp 461–463

DOI: 10.1021/op200354f

Development of a Robust Procedure for the Copper-catalyzed Ring-Opening of Epoxides with Grignard Reagents

Mahbub Alam, Christopher Wise, Carl A. Baxter, Ed Cleator, and Andrew Walkinshaw

Org. Process Res. Dev., 2012, 16 (3), pp 435–441

DOI: 10.1021/op200329x

Optimization Studies on the Hydro-acylation of 1-Alkenes to α-Methylketones using a Homogeneous Palladium/Josiphos Catalyst

Hans Heeres, Adri J. Minnaard, Bart Hessen, and Hero J. Heeres

Org. Process Res. Dev., 2012, 16 (3), pp 400–408

DOI: 10.1021/op100342v

Kilogram-Lab-Scale Oxindole Synthesis via Palladium-Catalyzed C–H Functionalization

E. Jason Kiser, Javier Magano, Russell J. Shine, and Michael H. Chen

Org. Process Res. Dev., 2012, 16 (2), pp 255–259

DOI: 10.1021/op200332p

A New Efficient Synthetic Route for the Synthesis of the Antiallergic Drug, Olopatadine Hydrochloride, via Stereospecific Palladium-Catalyzed Reaction

Koichiro Nishimura and Masahiko Kinugaw

Org. Process Res. Dev., 2012, 16 (2), pp 225–231

DOI: 10.1021/op200312m

Pd- and Mo-Catalyzed Asymmetric Allylic Alkylation

Barry M. Trost

Org. Process Res. Dev., 2012, 16 (2), pp 185–194

DOI: 10.1021/op200294r

Catalytic Hydrogenation of Esters. Development of an Efficient Catalyst and Processes for Synthesising (R)-1,2-Propanediol and 2-(l-Menthoxy)ethanol

Wataru Kuriyama, Takaji Matsumoto, Osamu Ogata, Yasunori Ino, Kunimori Aoki, Shigeru Tanaka, Kenya Ishida, Tohru Kobayashi, Noboru Sayo, and Takao Saito

Org. Process Res. Dev., 2012, 16 (1), pp 166–171

DOI: 10.1021/op200234j

Process Intensification via Reaction Telescoping and a Preliminary Cost Model to Rapidly Establish Value

Aman A. Desai, Erich J. Molitor, and John E. Anderson

Org. Process Res. Dev., 2012, 16 (1), pp 160–165

DOI: 10.1021/op200270f

An Efficient, Direct Bis-ortho-chlorination of 4-(Difluoromethoxy)aniline and Its Application to the Synthesis of BMS-665053, a Potent and Selective P

Jianqing Li, Daniel Smith, Subramaniam Krishnananthan, Richard A. Hartz, Bireshwar Dasgupta, Vijay Ahuja, William D. Schmitz, Joanne J. Bronson, Arvind Mathur, Joel C. Barrish, and Bang-Chi Chen

Org. Process Res. Dev., 2012, 16 (1), pp 156–159

DOI: 10.1021/op2003198

Allylic Amines as Key Building Blocks in the Synthesis of (E)-Alkene Peptide Isosteres

Erin M. Skoda, Gary C. Davis, and Peter Wipf

Org. Process Res. Dev., 2012, 16 (1), pp 26–34

DOI: 10.1021/op2002613