Assembly of Four Diverse Heterocyclic Libraries Enabled by Prins Cyclization, Au-Catalyzed Enyne Cycloisomerization, and Automated Amide Synthesis

Jiayue Cui, David I. Chai, Christopher Miller, Jason Hao, Christopher Thomas, JingQi Wang, Karl A. Scheidt, and Sergey A. Kozmin

J. Org. Chem., 2012, 77 (17), pp 7435–7470

DOI: 10.1021/jo301061r